Docking , Synthesis and Biological Evaluation of Novel Pyrazole, Pyrimidine and Thiazole derivatives attached to Naphthalene moiety as Cytotoxic and Antimicrobial agents

Faculty Pharmacy Year: 2015
Type of Publication: ZU Hosted Pages:
Authors:
Journal: World Journal of Pharmaceutical Research SJIF Impact Factor 5.990 Volume 4, Issue 7, 73-99. World Journal of Pharmaceutical Research SJIF Impact Factor 5.990 Volume 4, Issue 7, 73-99. Volume:
Keywords : Docking , Synthesis , Biological Evaluation , Novel Pyrazole,    
Abstract:
In the present study novel N-thiocarbamoyl pyrazole derivatives 2a-d and 3,4-dihydro pyrimidne-2(1H)-thione derivatives 3a-d were synthesized starting from α,β-unsaturated ketones 1a-d via reaction with thiosemicarbazide and thiourea respec
   
     
 
       

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