Click reaction based synthesis, antimicrobial, and cytotoxic activities of new 1,2,3-triazoles

Faculty	Science	Year:	2015
Type of Publication:	ZU Hosted	Pages:
Authors:	Hossam Aly Hussein Saad Staff Zu Site Abstract In Staff Site
Journal:	Bioorganic & Medicinal Chemistry Letters Elsevier Ltd.	Volume:

Keywords :	Click reaction based synthesis, antimicrobial, , cytotoxic
Abstract:	Three-motif pharmacophoric models 20a–e and 21–25 were prepared in good yields by CuAAC of two azido substrates 2 and 11 with seven terminal acetylenic derivatives including chalcones 17a–e, theo- phylline 18 and cholesterol 19. The structu

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