SYNTHESIS AND EVALUATION OF 2, 3-DIHYDROQUINAZOLIN-4(1H)-ONE DERIVATIVES AS ANALGESIC AND ANTI-INFLAMMATORY AGENTS

Faculty Pharmacy Year: 2013
Type of Publication: ZU Hosted Pages:
Authors:
Ahmed Samy Abdelsamad Abdelkhalek hilal
Journal: Asian Journal of Research in Chemistry and Pharmaceutical Sciences. international Volume:
Keywords : SYNTHESIS , EVALUATION , , 3-DIHYDROQUINAZOLIN-4(1H)-ONE DERIVATIVES , ANALGESIC , ANTI-INFLAMMATORY AGENTS    
Abstract:
Applying internal Mannich reaction on N'-(substituted benzoyl)-2-(methyl- amino) benzohydrazide (IIa-h), under different conditions, afforded a new series of 2, 3-dihydroquinazolin-4(1H)-one derivatives (IIIa-g). The carbohydrazide; N'-(p
    
     
 
       

Author Related Publications

  • Ahmed Samy Abdelsamad Abdelkhalek hilal, "Synthesis and biological screening of new derivatives of 2,3-dihydro quinazolin-4(1H)-one and benzotriazepin- 5(2H)-one for central nervous system activity", international, 2014 More
  • Ahmed Samy Abdelsamad Abdelkhalek hilal, "“Methylene Bridge” to 5-HT3 Receptor Antagonists Conformationally Constrained Phenylguanidines", American Chemical Society, 2018 More
  • Ahmed Samy Abdelsamad Abdelkhalek hilal, "Probing of 2-Amino-6-Chloro-3,4-Dihydroquinazoline Hydrochloride At 5- HT3 Receptor", Scholars Research Library, 2018 More
  • Ahmed Samy Abdelsamad Abdelkhalek hilal, "Probing of 2-Amino-6-Chloro-3,4-Dihydroquinazoline Hydrochloride At 5- HT3 Receptor", Scholars Research Library, 2018 More
  • Ahmed Samy Abdelsamad Abdelkhalek hilal, "X-ray crystal structure of a 2-amino-3, 4-dihydroquinazoline 5-HT3 serotonin receptor antagonist and related analogs", international, 2020 More

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